I-Indomethacin iyisidakamizwa esitholakala emafomu ahlukahlukene ekusetshenzisweni kwendawo nesistimu, kuhlanganise ngesimo samathebulethi. Ake sicabangele ngokuningiliziwe, yiziphi izibalo ezinikezwa amaphilisi anikeziwe, njengoba asebenza, yikuphi ukuphikisana kanye nemiphumela ababa nayo.
Ukwakhiwa kanye nezakhiwo zamakhemikhali amaphilisi Indomethacin
Isidakamizwa singeqembu lama-non-steroidal anti-inflammatory and antirheumatic drugs. Njengengxenye eyinhloko, iqukethe into efana negama elifanayo, okuyi-derivative ye-indoleacetic acid. Njengezithako ezengeziwe, amaphilisi, kuye ngokuthi umkhiqizi, angaqukatha: isitashi, i-silicon dioxide, i-lactose, i-talc, i-cellulose, i-lauryl sulfate, njll. Amaphilisi ahlanganiswe ne-enteric yembatho evimbela ukuchithwa kwesidakamizwa esiswini.
Izakhiwo zomzimba zalesi sidakamizwa zinjengalezi:
- anti-inflammatory;
- i-anesthetizing;
- antipyretic.
Lezi zindlela zokwelashwa zibangelwa ukuvimbela i-cyclooxygenase ye-enzyme, equkethe izicubu ezihlukahlukene zomzimba futhi inesibopho sokuhlanganiswa kwe-prostaglandins. I-Prostaglandin ibangela ubuhlungu ekugxilweni kwe-inflammation, ukwanda kwezinga lokushisa nokukhuphuka ekuphepheni kwamathambo; ngenxa yalokho, ngenxa yokunciphisa ukuhlanganiswa kwazo, lezi zimpawu ziyasuswa.
Isidakamizwa sinomthelela ekwehleni noma ekuqedeni ubuhlungu be-syndrome e-rheumatic non-rheumatic nature, okubandakanya kuthinta ubuhlungu obuhlangene ekuphumuleni nangomsebenzi. Futhi, kunciphisa ukuqina komzimba, kukhulisa umthamo wokunyakaza, ukulwa nokuvuvukala.
Izinkomba zokusebenzisa amaphilisi Indomethacin
Lawa amaphilisi anqunyelwe ukwelashwa ngokuphawulekayo kwezifo ezilandelayo:
- izifo ezivuthayo nezivuzayo zesimiso se-musculoskeletal (isifo samathambo, isifo sikaBeacherew, isifo sikaReiter, i-arthritis e-gouty, i-psoriatic arthritis, njll);
- izilonda zezicubu zesikhashana (bursitis, tendonitis, tendovaginitis, njll);
- ubuhlungu ngenxa yezilonda ezibuhlungu kanye nokuphathwa kokuhlinzwa;
- ukungahloniphi;
- i-radiculoneuritis;
- i-plexite;
- i-dysmenorrhea;
- i-adnexitis ;
- Izifo ezithathelwanayo nezivuthayo ezithombeni ze-ENT, njll.
Amathebulethi athathwa emva kokudla noma ngesikhathi saso emithini ngayinye, kuye ngokuthi uhlobo lwesifo nokuqina kwalo.
Imiphumela emibi ye-indomethacin
Lapho ukwelashwa kwe-Indomethacin kumathebulethi, izenzakalo ezimbi ezilandelayo zingase zenzeke:
- isicasuli;
- ubuhlungu besisu;
- ukuhlanza;
- izinkinga zesitoreji;
- ikhanda;
- ukuphuma kwegazi emaphethelweni emathunjini;
- ukulala;
- ukwanda kwengcindezi yegazi;
- ukuphazamiseka kwenhliziyo;
- itching;
- i-urticaria;
- i-anemia ;
- umbono ongenakwenzeka;
- ukucasuka, njll.
I-Contraindications Tablets Indomethacin
Imithi ye-Indomethacin kumaphilisi awavunyelwe ezimweni ezinjalo:
- ukuxhunywa komuntu kwizingxenye ze-ejenti;
- ukuba khona ku-anamnesis yokusabela ku-acetylsalicylic acid noma ezinye izidakamizwa eziphikisanayo nezibonakaliso zokuhlaselwa kwe-asthmatic, i-angioedema, i-hives, i-rhinitis;
- i-peptic ulcer;
- ukutholakala komlando wokugaya kwamathumbu noma ukugcoba ngenxa yokusetshenziswa kwesidakamizwa esingenalo isifo sokuvuvukala;
- ukwehluleka kwenhliziyo;
- isibindi esinzima noma ukwehluleka kwezinso;
- ukukhulelwa;
- isikhathi se-lactation.
Ngesikhathi ukwelashwa nge-indomethacin, kunconywa ukuqapha isibindi nezinso, ukubala kwegazi.