I-benzylpenicillin usawoti ka-sodium iyinhlanganisela eyinsawoti ye -sodium ye-benzylpenicillic acid, eyenziwa yizinhlobo ezithile ze-mold fungus. Lesi sidakamizwa singokomuthi we-antibiotics wechungechunge le-penicillin.
Ifomu lokukhiqizwa kwe-benzylpenicillin usawoti sodium
Isidakamizwa siyiphunga elihle, elenzelwe ukhiqiza isisombululo. I-benzylpenicillin usawoti ka-sodium ikhiqizwa ngezigxobo eziyizinkulungwane eziyi-1,000,000 - 100,000 zezinto ezisebenzayo. Izixazululo zezidakamizwa zisetshenziselwa imiphumela yesistimu emzimbeni (ngokuvamile okuyi-intramuscularly), imiphumela ezithombeni nasezicukwaneni ezidalwa yizidakamizwa ngegazi, futhi njengendlela yokuchayeka kwendawo. I-benzylpenicillin usawoti ka-sodium ayisetshenziswa ngomlomo, ngoba kubhujiswa kalula yisenzo sejusi esiswini.
Indlela yokusebenza ka-benzylpenicillin usawoti sodium
Isidakamizwa sinomthelela we-bactericidal kuma-microorganisms ezibucayi, ezisesiteji sokukhiqiza, futhi asithinti amangqamuzana aphumule. Ngesikhathi esifanayo, amabhaktheriya angenawo ama-intracellularly, futhi umphumela we-bactericidal uyabonakala ngisho nasezindlini eziphansi kakhulu ezidakamizwa.
I-benzylpenicillin usawoti ka-sodium ngemuva kokujova kwe-intramuscular ngokushesha ingena egazini, lapho iqhubekela khona ezingxenyeni zangaphakathi, izicubu neziphuzo futhi ihlala khona isikhathi eside. Eziningi kakhulu, lesi sidakamizwa sitholakala ezinso, isibindi, amaphaphu, i-lymph nodes, i-spleen, ezingxenyeni eziphansi - ezicubu ze-muscle, ama-pancreas, isikhumba se-thyroid, isikhumba. Ukungenwa kabi kwesidakamizwa ku-cartilage ne-bone tishu, i-cerebrospinal fluid.
Le antibiotic isebenza ngokumelene nama-microorganisms alandelayo:
- Ama-bacteria ama-Gram-positive (i-pneumococci, i-streptococci, i-staphylococci, i-diphtheria-pathogens, njll);
- I-gram-negative microbes (i-gonococci, i-meningococci);
- izinti ze-anaerobic ezenziwe nge-spore;
- i-spirochaetes;
- actinomycetes nezinye.
Ukuphikisana nesenzo se-benzylpenicillin usawoti ka-sodium kukhona ama-microorganisms ama-gram-negative (klebsiella, brucella), rickettsia, i-protozoa, amagciwane, cishe wonke ama-fungus, kanye nezinhlobo ze-staphylococci ezenza i-enzyme penicillinase. Umsebenzi onamandla uyabonakala ngokuphathelene namagciwane omzimba kanye nePseudomonas aeruginosa .
Ukusetshenziswa kosawoti ka-benzylpenicillin sodium
Ngokuvamile, lesi sidakamizwa sinqunywe ukwelashwa kwezifo ezincane zokuphefumula, izifo ezilimala, izifo zezingxenye ze-ENT, izifo ze-genitourinary, i-endocarditis ye-septic, izifo zamehlo, i-syphilis, ukuvuvukala kwentambo yomgogodla nobuchopho nezinye izifo ezibangelwa ama-microbes ezibucayi.
Isikhathi sokwelashwa sinqunywa uhlobo kanye nenkambo ye-pathology. Uma emva kwezinsuku ezimbili kuya kwezingu-3 emva kokuqala kokwelashwa akukho mphumela, bashintsha ekusetshenzisweni kwamanye ama-antibiotic.
Ungayinciphisa kanjani u-benzylpenicillin usawoti sodium?
Ukukhishwa kwe-benzylpenicillin usawoti sodium kwenziwa ngokushesha ngaphambi kokusetshenziswa. Ngomjovo we-intramuscular, intracavitary ne-subcutaneous, isidakamizwa sihlanjululwa ngamanzi for injection, saline noma isixazululo se-novocaine.
Ukujola kwe-jet engxenyeni ye-benzylpenicillin, usawoti we-sodium uchitheka emanzini ngenhloso yokujola noma isisindo saline. Ngaphambi kokusungulwa kokungena kwe-intravenous, lesi sidakamizwa sihlanjululwe ngesisombululo seglucose noma isisombululo saline. Ukuphathwa kwe-Endolumbral futhi
Ukusetshenziswa kwe-inhalation, i-benzylpenicillin powder of the sodium sodium incibilikiswe emanzini acwecwe noma isisombululo se-saline.
Ukungafani kwe-benzylpenicillin usawoti sodium:
- ukuzwela okukhulu ku-benzylpenicillin, kanye nezinye izidakamizwa ezivela eqenjini lama-penicillin ne-cephalosporin;
- isithuthwane (ukuphathwa kwe-endolumbral);
- ukukhulelwa kanye nokulahlwa;
- ukusabela okubi kakhulu kwe-allergic.