Ngokuvamile, abesifazane abahlushwa ukuhlaselwa ikhanda eliyingozi, bathatha ama- analgesics , okwenza ngcono isimo, futhi ekugcineni bayeke ukusiza. I-Triptans esuka ku-migraine iphumelela ngempela - izidakamizwa ezenzelwe ukuphatha lesi sifo. Abagcini nje ukukhulula ngokushesha ubuhlungu be-syndrome, kodwa nokuvimbela ukuthuthukiswa kokuhlaselwa, uma uthatha imithi kanye nezimpawu zokuqala ze-pathology.
Izidakamizwa ezivela eqenjini le-triptane zisebenza kanjani?
Indlela eyinhloko yomsebenzi waloluhlobo lwezidakamizwa ukugqugquzela ama-receipt of the walls of vascular. Ngaphezu kwalokho, i-tryptans ikhiqiza umphumela wokukhetha futhi usebenze kuphela ngaphakathi kwesikhashana, ngaphandle kokuphazamisa uhlelo lokujikeleza kwe-coronary and peripheral. Ngenxa yalokho, imithwalo yegazi egxilile ngokweqile, eyenza ukuba kunciphise masinyane ubuhlungu be-syndrome yobuhlungu.
Ngaphezu kwalokho, izidakamizwa ezichazwe zinciphisa ubuzwe bezintathu zokuthola izintathu ezingeni le-nucleus yomgogodla. Ngenxa yalolu buhlungu cishe aluzwa.
Ngaphezu kokuphathwa okusheshayo kwezimpawu ze- migraine , kuhlanganise ne-nausea, ukukhanya nomsindo, isizungu, imithi yeli qembu isetshenziselwa ukuvimbela. Ngokunciphisa ukuvuvukala kwe-neurogenic futhi kuvimbele ukungena emithanjeni yegazi.
I-Triptans inezinzuzo eziningana ngaphezu kwe-analgesics evamile:
- kubangele imiphumela emibi kakhulu;
- Ungabhubhisi umlutha kanye nesidingo sokwandisa umthamo;
- sebenze kunoma yisiphi isigaba sokuhlaselwa;
- ukuvimbela ukuqhubeka kobuhlungu, uma uthatha iphilisi ngezibonakaliso zokuqala;
- ukukhulula izimpawu ze-aura;
- ukulwa nemibonakaliso emtholampilo yesifo.
Yiziphi izidakamizwa ezihlobene nama-triptan?
Izidakamizwa ezibuzwayo zikhetha abaphikisi be-5HT18 / D. Ziyi-derivatives yamakhemikhali e-5-hydroxytryptamine, edingeka ngegama.
Kunezizukulwane ezimbili zezidakamizwa ezinama-triptan. Okokuqala kuhlanganisa yonke imishanguzo esekelwe ku-sumatriptan - ummeleli weqembu lokuqala. Isizukulwane sesibili sihlanganisa imithi enezithako ezilandelayo:
- zolmitriptan;
- eletriptan;
- i-naratriptan;
- i-almotriptan;
- rhizotriptan;
- lt; / RTI & gt;
Izidakamizwa ezintsha zithinta kakhulu imitholampilo kanye nezakhiwo ezithuthukisiwe zezokwelapha. Basiza ngokushesha futhi babangele imiphumela emibi kakhulu.
Kufanele kuqaphele ukuthi i-almo-, i-rhizo- kanye ne-fluorotriptans isayithola izivivinyo zezokwelapha futhi iyacwaninga, ngakho-ke ayitholakali mahhala.
Uhlu lwezidakamizwa ukusuka ku-migraine kusuka eqenjini lama-triptan
Ukuzithathela imithi yokwelashwa kungcono ngaphansi kokuboniswa udokotela. Naphezu kwendlela efanayo yesenzo se-triptans, isiguli ngasinye sisizwa uhlobo olulodwa lwemithi, oluzosiza ukhethe isazi ngemuva kokucwaninga ngokucophelela izici eziqondene nesiguli kanye ne-anamnesis.
Uhlu lwezidakamizwa:
1. Ama-Sumatriptans:
- Iphuzile;
- Imigran;
- Sumatriptan;
- Trimigrene;
- Amigrenin;
- I-Sumygamren.
2. Zolmitriptans:
- I-Zomig.
3. Ama-Eletriptans:
- Ama-Relpaks.
4. I-Naratriptans:
- I-Naramig.
Cishe isigamu sabantu abahlushwa yi-migraine ukuhlaselwa ikhanda libuyele ezinyangeni ezimbili ngisho nemithi echazwe. Ngakho-ke, okungenani amahora amabili ngemuva kokuthatha i-tryptane, kuphakanyiswa ukuthatha enye ithebhulethi yomuthi. Kubalulekile ukuthi ungadluli umthamo onconywayo.